CAS
136647-02-4
Formulation
A solid
Purity
≥98%
MW
466,062
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
An inhibitor of Kv1.3 and Kv1.4 (IC50s = 0.28 and 0.17 µM, respectively); selective for Kv1.3 and Kv1.4 over Kv1.1-1.2 and Kv1.5-1.6 (IC50s = 2.9-70 µM), Kv3.1, -3.2, and -3.4 (IC50s = 11-127 µM), Kv4.2 (IC50 = 10 µM), and KCa3.1/IK (IC50 = >30 µM); inhibits phytohemagglutinin-induced proliferation and IL-2 production in T cells (IC50s = 2 and 2.9 µM, respectively)
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).