
CAS
1135242-13-5
Formulation
A crystalline solid
Purity
≥98%
MW
369,9
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A selective agonist of M1 mAChRs (Ki = 9.91 µM); selective for M1 over M2-M5 mAChRs (Kis = 21.4-50 µM in CHO cells); increases calcium mobilization and activates the ERK signaling pathway (EC50 = 1.6 and 37 µM, respectively, in CHO cells expressing human recombinant M1 receptors); reverses scopolamine-induced deficits in contextual fear conditioning in rats (10 mg/kg)
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).