CAS
85375-15-1
Formulation
A solid
Purity
≥98%
MW
371,90008
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A GAT1 inhibitor (IC50s = 0.13 and 0.64 µM for the human and rat transporters, respectively); selective for GAT1 over rat GAT2, human GAT3, and human BGT3 (IC50s = 550, 944, and 7,210 µM, respectively); inhibits GABA uptake in rat synaptosome preparations (IC50 = 341 nM); inhibits DMCM-induced seizures in mice (ED50 = 3.1 mg/kg)
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).