CAS
288150-92-5
Formulation
A crystalline solid
Purity
≥98%
MW
356,4
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A potent OX1R antagonist (Ki = 26.9 nM in a calcium mobilization assay); selective for OX1R over OX2R (Kds = 21.7 and 1,704 nM, respectively, in a radioligand binding assay); co-perfusion with human OX1R in rat ventral tegmental area inhibits OX1R-induced glutamate and dopamine elevations; reduces cocaine-seeking behavior in rats
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).