Synonyms: 2-Phenylethynesulfonamide|PFT-μ


CAS
64984-31-2
Formulation
A crystalline solid
Purity
≥98%
MW
181,2
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
An inhibitor of p53-mediated apoptosis, preventing p53 binding at the mitochondrial surface without affecting p53 transactivational activities; at 25 μM, pifithrin-μ reduces p53-mediated apoptosis triggered by nutlin; also interacts selectively with Hsp70, disrupting its association with many substrate proteins
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).