Norelgestromin
CAY-35243-10 10 mg
Synonyms: 17-desacetyl Norgestimate|BRN 4202099|Levonorgestrel oxime|RWJ 10553
Data Sheet: 
SDS:
SDS:
CAS
53016-31-2
Formulation
A solid
Purity
≥95%
MW
327,4605
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
An active metabolite of norgestimate; an agonist of the progesterone receptor and ERα (EC50s= 11.1 and 43.4 nM, respectively); an antagonist of the glucocorticoid and mineralocorticoid receptors (IC50s = 255 nM and 83.7 nM, respectively); selectively binds progestin receptors (IC50 = 4.61 nM for rabbit uterine receptors) over androgen receptors (IC50 = 222 nM for rat prostatic receptors); activates the androgen receptor in a transactivation assay in MDA-MB-231 cells expressing the human receptor
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).
