CAS
886047-22-9
Formulation
A crystalline solid
Purity
≥98%
MW
437,94446
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A positive allosteric modulator of the M2 and M4 mAChRs; binds to allosteric sites on M2 and M4 receptors (KBs = 1.8-3.4 μM; potentiates the activity of ACh, iperoxo, and oxotremorine M at human recombinant M2 and M4 receptors expressed in CHO cell membranes; exhibits allosteric agonism at M2 and M4 receptors (23.2 and 16.8%, respectively, of the maximal ACh response)
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).