CAS
699020-93-4
Formulation
A solid
Purity
≥98%
MW
321,01186
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A potent histamine H3 receptor agonist (Ki = 0.85 nM); selective for histamine H3 over histamine H4 receptors (Ki = 245 nM); inhibits cAMP-stimulated β-galactosidase transcription in SK-N-MC cells expressing human H3 receptors (EC50 = 0.18 nM); induces a decrease of the electrically induced twitch contraction in isolated guinea pig ileum; inhibits hydrochloric acid-induced formation of gastric lesions in rats at 30 mg/kg, s.c.
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).