CAS
2088410-46-0
Formulation
A solid
Purity
≥98%
MW
325,4
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A BET BD2 inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD3, BRD4, and BRDT BD2, respectively); selective for BD2 in BRD2, BRD3, BRD4, and BRDT over BD1 in the same BRDs (IC50s = >15,000 nM for all); inhibits LPS-induced CCL1 production in isolated human whole blood (IC50 = 794.3 nM)
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).