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PI(3)K-Akt-mTOR Pathway

   

  PI3-K, Akt/PKB, and mTOR - NEW!!


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PI3-K Enzymes / PI3-K Antibodies / PI3-K Peptides and Substrates / PI3-K Inhibitors
mTOR Antibodies / mTOR Inhibitor
Akt/PKB and p70 S6 Kinase Enzymes / Akt/PKB and p70 S6 Kinase Antibodies / Akt and p70 S6 Kinase Peptides and Substrates / Akt Inhibitors & Activators

 

Monoclonal and Polyclonal Antibodies

MAb to Akt (19G7), Mouse IgG1

ALX-803-303

MAb to Akt (5C10), Mouse IgG1

ALX-804-553

MAb to Akt (5C10), Mouse IgG1

NT-0119

MAb to AKT (8F4), Mouse IgG1

BML-SA312

MAb to AKT (dephosphorylated) (11A11), Mouse IgG1

BML-SA313

MAb to Akt (dephosphorylated) (11A11), Mouse IgG1

ALX-804-400

MAb to Akt (dephosphorylated) (Ser473) (11A11), Mouse IgG1

NT-0049

MAb to Akt1 (5G12), Mouse IgG1

ALX-804-633

MAb to Akt1 (5G12), Mouse IgG1

NT-0144

MAb to Akt2 (human) (8B7), Mouse IgG2a

ALX-804-634

MAb to Akt2 (human) (8B7), Mouse IgG2a

NT-0179

MAb to Akt3 (human) (66C1247.1), Mouse IgG1

ALX-804-379

MAb to PDK Substrate (phosphorylated) (2D2), Mouse IgG1

ALX-804-397

MAb to PDK Substrate (phosphorylated) (2D2), Mouse IgG1

NT-0056

MAb to PDK Substrate (phosphorylated) (4E1), Mouse IgG1

ALX-804-398

MAb to PDK Substrate (phosphorylated) (4E1), Mouse IgG1

NT-0057

MAb to Phosphoinositide 3-kinase p110γ (H1), Mouse IgG2a ALX-804-230
MAb to PI 3-Kinase (p85α Subunit) (8-2D-4D), Mouse IgG1 BML-SA269
MAb to PTEN (11G8.1), Mouse IgG ALX-804-451
MAb to PTEN (6H2.1), Mouse IgG ALX-804-254
MAb to Raptor (10E10), Mouse IgG1 NT-0255
MAb to Rictor (1G11), Mouse IgG1 NT-0250
MAb to αhPI(3)Kγ (641) JBS-ABD-027
MAb to αhPI(3)Kγ (641) JBS-ABD-027P
MAb to αhPI(3)Kγ (H1) JBS-ABD-026L
MAb to αhPI(3)Kγ (H1) JBS-ABD-026S
MAb to Akt (phosphorylated) (pSer473) (11E6), Mouse IgG1 ALX-804-401
MAb to Akt (phosphorylated) (pSer473) (11E6), Mouse IgG1 NT-0108
MAb to PIP2 (human) (2C11), IgM ABR-MA3-500
MAb to SHIP-1 (human) (SHIP-01) (Purified), Mouse IgG2a EXB-11-524
MAb to SHIP-1 (human) (SHIP-02) (Purified), Mouse IgG2a EXB-11-525
Monoclonal Antibody to Omentin 1 (human) (Saly-1), Mouse IgG2b ALX-804-850
Monoclonal Antibody to Omentin 1 (human) (Saly-2), Mouse IgG2a ALX-804-852
PAb to Akt (activated) (pSer473) BV-3257
PAb to Akt (phosphorylated) (pSer473), From rabbit. BML-SA450
PAb to Akt (phosphorylated) (pThr308), From rabbit. BML-SA290
PAb to Akt, From rabbit. ; anti-PKB PAb; anti-Protein Kinase B PAb ALX-210-226
PAb to Akt/PKB BV-3247
PAb to Akt1 (NT), From rabbit. PSC-3519
PAb to FKBP12 BV-3635
PAb to FKBP12, From rabbit.    ABR-PA1-026A
PAb to G Protein β Subunit-like PSC-3495
PAb to Inositol 1,4,5-trisphosphate Receptor (Type-I), From rabbit. ALX-210-115
PAb to Inositol 1,4,5-trisphosphate Receptor (Type-I), From rabbit. ALX-210-169
PAb to Inositol 1,4,5-Trisphosphate Receptor (Type-I), From rabbit.    ABR-PA1-901
PAb to Inositol 1,4,5-Trisphosphate Receptor (Type-I), From rabbit.    ABR-PA3-901A
PAb to Inositol 1,4,5-Trisphosphate Receptor (Type-II) (rat), From rabbit.    ABR-PA1-904
PAb to Inositol 1,4,5-trisphosphate Receptor (Type-II), From rabbit. ALX-210-224
PAb to Inositol Hexakisphosphate [IP6] Kinase (rat), From rabbit.    ABR-PA1-906
PAb to mTOR ABR-PA1-518
PAb to mTOR (human FRB Domain), From rabbit. ; anti-mTOR (human FKBP12-rapamycin-binding Domain) PAb ALX-215-065
PAb to mTOR (NT), From rabbit.  PSC-3485
PAb to mTOR  , From rabbit. ; anti-Mammalian Target of Rapamycin PAb; anti-FRAP1 PAb ALX-210-065
PAb to Omentin 1 (AT117), From rabbit. ALX-210-941
PAb to Omentin 1 (human), From rabbit. ALX-210-454
PAb to p70 S6 Kinase BV-3485
PAb to p70 S6 Kinase (activated) BV-3505
PAb to PDK1 BV-3449
PAb to PH Domain Leucine-rich Repeat Protein Phosphatase, From rabbit. CAY-10007191
PAb to PIKE (CT), From rabbit. PSC-3321
PAb to pp36 (human), From rabbit. ALX-210-770
PAb to PRAS40 (phosphorylated) (pThr246), From rabbit. BML-SA360
PAb to Protein Kinase B (mouse), From rabbit.    ABR-PA1-540
PAb to PTEN BV-3479
PAb to PTEN (CT), From rabbit. PSC-3515
PAb to PTEN (NT), From rabbit. PSC-3517
PAb to PTEN Induced Putative Kinase 1 (PINK1) CAY-10006283
PAb to PTEN, From rabbit. CAY-10005059
PAb to Raptor (IN), From rabbit. PSC-3493
PAb to Raptor (mouse) (CT) PSC-3489
PAb to Raptor (NT) PSC-3491
PAb to Ribosomal Protein S6 Kinase (70kDa) (human) (phosphorylated) (pThr389), From rabbit. ABR-PA1-526
PAb to Ribosomal Protein S6 Kinase 1 (human) (NT), From rabbit. PSC-3511
PAb to Ribosomal S6 Kinase 2 (rat), From rabbit. CAY-10009411
PAb to TSC1 (CT), From rabbit. PSC-3503
PAb to TSC1 (IN), From rabbit. PSC-3505
PAb to TSC2 (CT), From rabbit. PSC-3507
PAb to TSC2 (NT), From rabbit. PSC-3509
PAb to Akt1 (85-100) (human) (Purified), From rabbit. EXB-11-509
PAb to CARP, From rabbit. ABR-PA3-852
PAb to PTEN (human) (CT) (Purified), From rabbit. EXB-11-510
PAb to PTEN, From rabbit. ABR-PA1-808
PAb to WIPI-1 (AT130), From rabbit. ALX-210-955
PAb to WIPI-1 (human) (AT129), From rabbit. ALX-210-954
PAb to Akt (mouse), From rabbit. ALX-210-534
PAb to FKBP12, From rabbit. ALX-210-142
PAb to Inositol Hexakisphosphate Kinase (rat), From rabbit. ALX-210-289
PAb to Phosphatidylinositol-4-phosphate 5-kinase-Iγ, From rabbit. ALX-210-745
PAb to Phosphoinositide 3-Kinase p110δ (human), From rabbit. ALX-210-747
PAb to Ribosomal Protein S6 Kinase (70kDa) (human) (phosphorylated) (pThr389), From rabbit. ALX-210-068
PAb to Tribbles Homolog 3, From rabbit. CVL-PAB0406
Polyclonal Antibody to mTOR BV-3786
Polyclonal Antibody to TRB-3 (human), From rabbit. ALX-210-462
Recombinant Proteins  
Akt (human) (recombinant) Western Ready Control CAY-10010079
Akt1 (active) BV-7701
Akt1 (human) (recombinant) BML-SE260
Akt1 (human) (recombinant) BML-SE416
Akt1/ PKBαHis (human) (recombinant) (active) JBS-PR-324
Akt1/ PKBαHis, inactive JBS-PR-325
Akt2 (active) BV-7702
Akt2 (human) (recombinant) BML-SE247
Akt2 (human) (recombinant) (activated) BML-SE248
Akt2/PKBβHis (human) (recombinant) (active) JBS-PR-333
Akt3 (active) BV-7703
Akt3 (human) (recombinant) BML-SE369
Akt3/ PKBγHis (human) (recombinant) (active) JBS-PR-334
Omentin 1 (human) (recombinant) ALX-522-108
Omentin 1 (human) (recombinant) (His) ALX-201-371
Omentin (rat) (recombinant) ALX-522-132
p70 S6 Kinase (human) (recombinant) BML-SE345
P70 S6K (active) BV-7725
pCAF Histone Acetyltransferase (human) (recombinant) (GST) CAY-10009115
PDK1 (active) BV-7706
Phosphoinositide 3-kinase p110α/p85 (bovine) (recombinant) ALX-201-119
Phosphoinositide 3-kinase p110γ (human) (recombinant) ALX-201-055
Phosphoinositide 3-kinase p85α (Regulatory Subunit) (bovine) (recombinant) JBS-PR-342
PI3 Kinase (human) (recombinant) BML-SE436
PI3 Kinase α (bovine) (recombinant) JBS-PR-341
PI3 Kinase α GST (bovine) (recombinant) JBS-PR-940
PI3 Kinase α R916P GST (bovine) (recombinant) JBS-PR-941
PI3 Kinase βHis (human) (recombinant) JBS-PR-344
PI3 Kinase γ D946A GST (human) (recombinant) JBS-PR-346
PI3 Kinase γ His (human) (recombinant) JBS-PR-343
PI3 Kinase δ GST (human) (recombinant) JBS-PR-345
PRAS40 (human) (recombinant) BML-SE308
PtdIns-(3,4,5)-P3 Binding Protein (E.coli) (recombinant) (GST) CAY-10009817
PtdIns-(4)-P1 Binding Protein (E. coli) (recombinant) (GST) CAY-10009241
PtdIns-(4,5)-P2 Binding Protein (E. coli) (recombinant) (GST) CAY-10009815
PTEN (human) BV-4838
PTEN (human) (recombinant) BML-SE402
PTEN (human) (recombinant) (GST) Western Ready Control CAY-10009747
PTEN (human) (recombinant) (His) CAY-10009746
RSK1 (human) (recombinant) BML-SE429
RSK2 (recombinant) (active) BV-7768
RSK3 (recombinant) (active) BV-7774
Ship2 (human) (recombinant) BML-SE539
Assay Kits & Sets  
KinaseSTAR Akt Activity Assay Kit BV-K435
Omentin 1 (human) Detection Set [For ELISA Application] APO-54N-026
Omentin 1 (human) ELISA Kit APO-54N-034
PI3K Lipid Kinase Substrate Mix 1 JBS-LI-011
PI3K Lipid Kinase Substrate Mix 2 JBS-LI-012
TOR Signalling Pathway Detection Set PSC-PSI-1805
Substances  
(-)-Epigallocatechin gallate ALX-270-263
(+)-Xestospongin A CAY-10006794
()-Naringenin ALX-385-010
1,2-Di-O-butyryl-D-myo-inositol 3,4,5,6-tetrakisphosphate octakis(propionoxymethyl)ester ALX-307-063
1-D-3-Deoxy-phosphatidylinositol ALX-307-002
1L-6-Hydroxymethyl-chiro-inositol-2-[(R)-2-O-methyl-3-O-octadecylcarbonate] ALX-270-292
2,3-Di-O-butyryl-D-myo-inositol 1,4,5,6-tetrakisphosphate octakis(propionoxymethyl)ester ALX-307-060
2,5,6-Tri-O-butyryl-D-myo-inositol 1,3,4-trisphosphate hexakis(acetoxymethyl)ester ; Bt3Ins(1,3,4)P3/AM ALX-307-045
3-Deoxy-3-bromo-D-myo-inositol 1,4,5-trisphosphate . hexasodium salt ALX-307-018
3-Deoxy-3-fluoro-D-myo-inositol 1,4,5-trisphosphate . hexasodium salt ALX-307-021
6BIO ALX-430-156
Akt (pSer473) Control Peptide Pair BML-SP288
Akt (pThr308) Control Peptide Pair BML-SP290
Akt Inhibitor BV-1701
Akt Substrate BML-P129
AKT/PKB substrate peptide JBS-PE-200
Araguspongin B CAY-10006797
AS-252424
PI(3)K p110γ Isoform Selective Inhibitor. Potent and selective phosphoinositide 3-kinase (PI(3)K) p110γ inhibitor shown to be selective for class IB PI(3)K-mediated cellular effects. LIT: Sequential activation of class IB and class IA PI3K is important for the primed respiratory burst of human but not murine neutrophils: A.M. Condliffe, et al.; Blood 106, 1432 (2005) - Furan-2-ylmethylene thiazolidinediones as novel, potent, and selective inhibitors of phosphoinositide 3-kinase gamma: J. Med. Chem. 49, 3857 (2006)
ALX-270-465
AS-252424 CAY-10009052
AS-604850
PI(3)K p110γ Isoform Selective Inhibitor. Potent, cell permeable and ATP-competitive inhibitor of phosphoinositide 3-kinase (PI(3)K) p110γ. Exhibits selectivity over other PI(3)K isoforms. LIT: Blockade of PI3Kgamma suppresses joint inflammation and damage in mouse models of rheumatoid arthritis: M. Camps, et al.; Nat. Med. 11, 936 (2005) - Key role of the p110delta isoform of PI3K in B-cell antigen and IL-4 receptor signaling: comparative analysis of genetic and pharmacologic interference with p110delta function in B cells: A. Bilancio, et al.; Blood 107, 642 (2006)
ALX-270-461
AS-604850 CAY-10010175
AS-605240
PI(3)K p110γ Isoform Selective Inhibitor. Potent, cell permeable and ATP-competitive inhibitor of phosphoinositide 3-kinase (PI(3)K) p110γ. Exhibits selectivity over other PI(3)K isoforms. LIT: PI3Kgamma inhibition blocks glomerulonephritis and extends lifespan in a mouse model of systemic lupus: D.F. Barber, et al.; Nat. Med. 11, 933 (2005) - Blockade of PI3Kgamma suppresses joint inflammation and damage in mouse models of rheumatoid arthritis: M. Camps, et al.; Nat. Med. 11, 936 (2005)
ALX-270-462
AS-605240 CAY-10007707
Biotinylated-Crosstide BML-P191
BML-257 BML-EI336
CAY10567 CAY-10010233
Compound 15e ALX-270-455
Crosstide BML-P149
Deguelin BML-EI329
Deguelin ALX-350-118
DL-myo-Inositol 1,3,4,5-tetrakisphosphate . tetrapotassium salt ALX-307-032
DL-myo-Inositol 1,4,5,6-tetrakisphosphate . tetrapotassium salt ALX-307-033
DL-myo-Inositol 1,5-bisphosphate . dipotassium salt ALX-307-027
D-myo-Inositol 1,2,3,4,5-pentakisphosphate . decasodium salt ALX-307-074
D-myo-Inositol 1,2,3,4,6-pentakisphosphate . decasodium salt ALX-307-075
D-myo-Inositol 1,2,3,4-tetrakisphosphate . tetrapotassium salt ALX-307-040
D-myo-Inositol 1,2,3,5,6-pentakisphosphate . decasodium salt ALX-307-076
D-myo-Inositol 1,2,3,5-tetrakisphosphate . tetrapotassium salt ALX-307-031
D-myo-Inositol 1,2,3,6-tetrakisphosphate . tetrapotassium salt ALX-307-041
D-myo-Inositol 1,2,3-trisphosphate . tripotassium salt ALX-307-042
D-myo-Inositol 1,2,4,5-tetrakisphosphate . octasodium salt ALX-307-053
D-myo-Inositol 1,3,4,5,6-pentakisphosphate . pentapotassium salt ALX-307-037
D-myo-Inositol 1,3,4,5-tetrakisphosphate . tetrapotassium salt ALX-307-005
D-myo-Inositol 1,3,4-trisphosphate . hexapotassium salt ALX-307-006
D-myo-Inositol 1,3,5,6-tetrakisphosphate . tetrapotassium salt ALX-307-036
D-myo-Inositol 1,3,5-trisphosphate . hexasodium salt ALX-307-047
D-myo-Inositol 1,3,6-trisphosphate . hexasodium salt ALX-307-050
D-myo-Inositol 1,4,5,6-tetrakisphosphate . tetrapotassium salt ALX-307-034
D-myo-Inositol 1,4,5-trisphosphate (caged) . trisodium salt ALX-307-070
D-myo-Inositol 1,4,5-trisphosphate . hexapotassium salt ALX-307-007
D-myo-Inositol 1,4,5-trisphosphate . hexasodium salt ALX-307-009
D-myo-Inositol 1,4,5-trisphosphate . triammonium salt ALX-307-011
D-myo-Inositol 1,4,5-trisphosphate . trilithium salt ALX-307-013
D-myo-Inositol 1,4,6-trisphosphate . tripotassium salt ALX-307-029
D-myo-Inositol 1,5,6-trisphosphate . tripotassium salt ALX-307-043
D-myo-Inositol 1,5-bisphosphate . tetrapotassium salt ALX-307-028
D-myo-Inositol 1-monophosphate . dipotassium salt ALX-307-026
D-myo-Inositol 2,3,4,5,6-pentakisphosphate . decasodium salt ALX-307-077
D-myo-Inositol 2,3,5-trisphosphate . tripotassium salt ALX-307-030
D-myo-Inositol 3,4,5,6-tetrakisphosphate . octasodium salt ALX-307-061
D-myo-Inositol 3,4,5-trisphosphate . tripotassium salt ALX-307-044
D-myo-Inositol 3,4,5-trisphosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-079
D-myo-Inositol 3,4,6-trisphosphate . hexasodium salt ALX-307-073
D-myo-Inositol 3,4-bisphosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-038
D-myo-Inositol 3-monophosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-080
D-myo-Inositol 4,5-bisphosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-039
D-myo-Inositol 4-monophosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-081
D-myo-Inositol 5-monophosphate, L-α-Phosphatidyl-(1,2-dipalmitoyl)- ALX-307-082
D-myo-Inositol-1,2,3,4-tetraphosphate . sodium salt CAY-10008448
D-myo-Inositol-1,2,3,5-tetraphosphate . sodium salt CAY-10008449
D-myo-Inositol-1,2,3,5-tetraphosphate . sodium salt CAY-10008451
D-myo-Inositol-1,2,3,6-tetraphosphate . sodium salt CAY-10008450
D-myo-Inositol-1,2,4,5,6-pentaphosphate . sodium salt CAY-10008452
D-myo-Inositol-1,2,5,6-tetraphosphate . sodium salt CAY-10008444
D-myo-Inositol-1,2,6-triphosphate . sodium salt CAY-10007780
D-myo-Inositol-1,2-diphosphate . sodium salt CAY-10008439
D-myo-Inositol-1,3,4,5,6-pentaphosphate . ammonium salt CAY-10009851
D-myo-Inositol-1,3,4,5,6-pentaphosphate . sodium salt CAY-10007784
D-myo-Inositol-1,3,4,6-tetraphosphate . ammonium salt CAY-10008442
D-myo-Inositol-1,3,4-triphosphate . sodium salt CAY-60972
D-myo-Inositol-1,3,5-triphosphate . sodium salt CAY-10007781
D-myo-Inositol-1,3-diphosphate . sodium salt CAY-10008443
D-myo-Inositol-1,4,5,6-Tetraphosphate . sodium salt CAY-10007783
D-myo-Inositol-1,4,5-triphosphate . hexapotassium salt BML-CA430
D-myo-Inositol-1,4,5-triphosphate . hexasodium salt BML-CA435
D-myo-Inositol-1,4,5-triphosphate . sodium salt CAY-10008205
D-myo-Inositol-1,4,5-triphosphate . trilithium salt BML-CA440
D-myo-Inositol-1,4,5-triphosphate . potassium salt CAY-60960
D-myo-Inositol-1,4,6-triphosphate . sodium salt CAY-10008427
D-myo-Inositol-1,4-diphosphate . sodium salt CAY-10008438
D-myo-Inositol-1,5-diphosphate . sodium salt CAY-10008441
D-myo-Inositol-1-phosphate . sodium salt CAY-10007777
D-myo-Inositol-2,3,4,5-tetraphosphate . ammonium salt CAY-10008456
D-myo-Inositol-2,3,5-triphosphate . ammonium salt CAY-10008423
D-myo-Inositol-2,4,5-triphosphate . sodium salt CAY-10007779
D-myo-Inositol-2,5,6-triphosphate . sodium salt CAY-10008424
D-myo-Inositol-3,4,5,6-tetraphosphate . sodium salt CAY-10007782
D-myo-Inositol-3,4,5-triphosphate . sodium salt CAY-10008425
D-myo-Inositol-3-phosphate . sodium salt CAY-10007778
D-myo-Inositol-4,5-diphosphate . sodium salt CAY-10008418
D-myo-Inositol-4-phosphate . ammonium salt CAY-10008437
Epigallocatechin Gallate CAY-70935
Epigallocatechin gallate LKT-E6234
Fumonisin B1 ALX-350-017
Gambogic amide BML-N159
H-89 CAY-10010556
H-89 . 2HCl BML-EI196
H-89 . dihydrochloride ALX-270-017
Inositol LKT-I5357
iso-Ins(1,4,5)P3/PM (caged) ALX-307-071
L-Quebrachitol ALX-307-001
Luteolin ALX-385-007
Luteolin CAY-10004161
Luteolin LKT-L8377
LY 294002 BML-ST420
LY-294,002 Bulk!
Potent, cell permeable inhibitor of phosphoinositide 3-kinase (PI(3)K) that acts on the ATP binding site of the enzyme.
ALX-270-038
LY294002 CAY-70920
LY294002 JBS-INH-002
LY-303,511  Bulk!
Useful negative control for the PI(3)K inhibitor LY-294,002 (Prod. No. ALX-270-038).
Does not inhibit phosphoinositide 3-kinase (PI(3)K) even at concentrations ≥100μM (LY-294,002: IC50=1.4μM).
ALX-270-410
L-α-Phosphatidylinositol BML-PH100
L-α-Phosphatidylinositol-3,4,5-P3 BML-PH107
L-α-Phosphatidylinositol-3,4-P2 BML-PH106
L-α-Phosphatidylinositol-3-P BML-PH105
L-α-Phosphatidylinositol-4-P BML-PH101
ML-9 BML-EI153
ML-9 CAY-10010236
myo-Inositol ALX-307-003
Myo-inositol galactoside MGT-M0326
N-Acetyl-Asp-Tyr(2-malonyl)-Val-Pro-Met-Leu-NH2 ALX-151-026
N-Acetyl-Asp-Tyr(PO3H2)-Val-Pro-Met-Leu-NH2 ALX-151-027
NaD-myo-Inositol-1,3,4,5-tetraphosphate . sodium salt CAY-60980
N-Arachidonoyl-L-serine ALX-340-063
N-Arachidonoyl-L-serine CAY-10005455
Naringenin LKT-N0068
PAK4/AKT Peptide Substrate BML-P194
Paxilline ALX-630-019
Paxilline LKT-P0392
PI JBS-LI-001
PI JBS-LI-008
PI-103
PI(3)K Inhibitor with an Interesting Profile. Potent, cell permeable and ATP-competitive inhibitor of DNA-PK, phosphoinositide 3-kinase (PI(3)K), the rapamycin-sensitive (mTORC1) and rapamycin-insensitive (mTORC2) complexes of the protein kinase mTOR. Exhibits little activity towards a panel of more than 40 other kinases even at concentrations as high as 10μM. Effectively blocks cell proliferation in glioma cell lines both in vitro and in vivo. LIT: A dual PI3 kinase/mTOR inhibitor reveals emergent efficacy in glioma: Q.W. Fan, et al.; Cancer Cell 9, 341 (2006) - A pharmacological map of the PI3-K famisly defines a role for p110alpha in insulin signaling: Z.A. Knight, et al.; Cell 125, 733 (2006)
ALX-270-460
PI-103 CAY-10009209
PI3-Kinase α Inhibitor 2 CAY-10010177
PI-4,5-P2 JBS-LI-003
PI-4,5-P2 JBS-LI-010
PI-4-P JBS-LI-002
PI-4-P JBS-LI-009
PKC412 ALX-380-281
PLC Thio-PIP2 . sodium salt CAY-10007839
PRAS40 (pThr246) Control Peptide Pair BML-SP360
Ptd(S)Ins-(3,4)-P2 (1,2-dioctanoyl) . sodium salt CAY-10010181
Ptd(S)Ins-(3,4)-P2 (1,2-dipalmitoyl) . sodium salt CAY-10010112
PtdIns-(1,2-dioctanoyl) . sodium salt CAY-10008099
PtdIns-(1,2-dipalmitoyl) .  ammonium salt CAY-10007710
PtdIns-(3)-P1 (1,2-dioctanoyl) . sodium salt CAY-10008394
PtdIns-(3)-P1 (1,2-dipalmitoyl) (triammonium salt) CAY-64921
PtdIns-(3)-P1 (1,2-dipalmitoyl)-d62 . ammonium salt CAY-10005616
PtdIns-(3,4)-P2 (1,2-dihexanoyl) . sodium salt CAY-10007759
PtdIns-(3,4)-P2 (1,2-dioctanoyl) . sodium salt CAY-10008400
PtdIns-(3,4)-P2 (1,2-dipalmitoyl) CAY-64922
PtdIns-(3,4,5)-P3 (1,2-dioctanoyl) . sodium salt CAY-10007764
PtdIns-(3,4,5)-P3 (1,2-dipalmitoyl) CAY-64920
PtdIns-(3,4,5)-P3 (1-stearoyl, 2-arachidonyl) CAY-64930
PtdIns-(3,4,5)-P3-biotinamide . sodium salt CAY-10009531
PtdIns-(3,4,5)-P3-fluorescein . triethylammonium salt CAY-10010383
PtdIns-(3,5)-P2 (1,2-dihexanoyl) . sodium salt CAY-10008396
PtdIns-(3,5)-P2 (1,2-dioctanoyl) . sodium salt CAY-10007763
PtdIns-(3,5)-P2 (1,2-dipalmitoyl) . trisodium salt CAY-10008398
PtdIns-(4)-P1 (1,2-dihexanoyl) . sodium salt CAY-10007757
PtdIns-(4)-P1 (1,2-dioctanoyl) . ammonium salt CAY-10007711
PtdIns-(4)-P1 (1,2-dipalmitoyl) CAY-64923
PtdIns-(4,5)-P2 (1,2-dihexanoyl) . sodium salt CAY-10007762
PtdIns-(4,5)-P2 (1,2-dioctanoyl) CAY-64910
PtdIns-(4,5)-P2 (1,2-dipalmitoyl) CAY-64924
PtdIns-(4,5)-P2 (1,2-dipalmitoyl) . sodium salt CAY-10008115
PtdIns-(4,5)-P2 (1,2-dipalmitoyl)-d62 . sodium salt CAY-10005615
PtdIns-(4,5)-P2-biotinamide . sodium salt CAY-10008159
PtdIns-(4,5)-P2-fluorescein . triethylammonium salt CAY-10010388
PtdIns-(5)-P1 (1,2-dihexanoyl) . sodium salt CAY-10008050
PtdIns-(5)-P1 (1,2-dioctanoyl) . ammonium salt CAY-10007758
PtdIns-(5)-P1 (1,2-dipalmitoyl) CAY-64925
Rapamycin ALX-380-004
Rapamycin BML-A275
Rapamycin BV-1568
Rapamycin LKT-R0161
S6 Peptide BML-P116
S6 Ribosomal Protein/Peptide BML-P144
S6-1 LKT-S0006
scyllo-Inositol ; Scyllitol ALX-307-004
SH-5 ALX-270-349
SH-6 ALX-270-350
TG 100-115 CAY-10010512
TGX-221 ALX-270-464
TGX-221
PI(3)K p110β Isoform Selective Inhibitor. Potent, selective and cell permeable inhibitor of phosphoinositide 3-kinase (PI(3)K) p110β. LIT: Sequential activation of class IB and class IA PI3K is important for the primed respiratory burst of human but not murine neutrophils: A.M. Condliffe, et al.; Blood 106, 1432 (2005) - PI 3-kinase p110beta: a new target for antithrombotic therapy: S.P. Jackson, et al.; Nat. Med. 11, 507 (2005)
CAY-10007349
Triciribine BML-EI332
Triciribine CAY-10010237
Wortmannin ALX-350-020
Wortmannin BML-ST415
Wortmannin CAY-10010591
Wortmannin LKT-W5769
Xestospongin C ALX-350-382
Xestospongin C BML-CA409
Xestospongin C CAY-64950
ZSTK474
PI(3)K Inhibitor with Antitumor Activity. Cell permeable, reversible, potent and specific inhibitor of phosphoinositide 3-kinase (IC50=17nM for PI(3)K p110β, IC50=53nM for PI(3)K p110γ and IC50=6nM for PI(3)K p110δ). Blocks cellular PI(3)K/Akt signalling in vitro and inhibits Akt-dependent tumor growth in mice in vivo without significant toxic effect. More effective than LY-294,002 (Prod. No. ALX-270-038) in vitro and in vivo. LIT: A novel phosphatidylinositol 3-kinase inhibitor, ZSTK474 exerted antitumor activity against human tumor xenografts by oral administration: S.Yaguchi et al.; Proc. Am. Assoc. Cancer Res. 46, 1691 (2005) - Antitumor activity of ZSTK474, a new phosphatidylinositol 3-kinase inhibitor: S. Yaguchi, et al.; J. Natl. Cancer Inst. 98, 545 (2006) Not sold in USA & Japan
ALX-270-454

    



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